Detailed definition
Gabapentin, originally developed as an anticonvulsant, is structurally similar to GABA but acts primarily on voltage-gated calcium channels rather than GABA receptors. Multiple RCTs show modest reductions in hot flash frequency (roughly 25–45%) at doses of 300–900 mg/day, with the strongest evidence for nighttime dosing reducing night sweats and improving sleep. Side effects include daytime sedation, dizziness, and weight gain. Pregabalin (Lyrica) has similar effects with a smaller evidence base.
Why it matters in menopause
For women whose dominant menopause complaint is nighttime hot flashes that destroy sleep — and who cannot or do not want to use estrogen — bedtime gabapentin is a useful option. Many menopause practices use it as a sleep-VMS combined intervention.
Related terms
Sources
External references: Wikipedia.