Glossary · Treatments

Clonidine

Definition: Clonidine is a centrally-acting alpha-2 adrenergic agonist originally developed for hypertension. It has modest efficacy for hot flashes (roughly 15–30% reduction) and is rarely first-line, but remains an option for women who cannot use estrogen, SSRIs/SNRIs, or fezolinetant.

Detailed definition

Clonidine is an alpha-2 adrenergic agonist that reduces sympathetic outflow. For vasomotor symptoms, evidence shows a modest reduction in hot flash frequency (roughly 15–30%), notably less than HRT, fezolinetant, or paroxetine. It is available as oral tablets or transdermal patches. Side effects include hypotension, dizziness, dry mouth, sedation, and rebound hypertension on discontinuation. It is rarely first-line for VMS in modern practice but is occasionally useful for women with concurrent hypertension or who cannot use other options.

Why it matters in menopause

Clonidine has a small remaining role for women who are not candidates for estrogen, SSRIs/SNRIs, gabapentin, or fezolinetant. It is rarely the first choice but can fit specific clinical situations.

Sources

External references: Wikipedia.

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